SCHEMBL8690765

SCHEMBL8690765

CCc1c(-c2c(-c3cc(C)cc(C)c3)[nH]c3ccc(O)cc23)ccc2c1C(=O)NC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WEE1 P30291 17/20 0.50
CHEK1 O14757 14/20 0.50
ROCK2 O75116 2/20 0.42
MEN1 O00255 1/20 0.40
PRKD3 O94806 1/20 0.40
PRKCG P05129 1/20 0.40
PRKCB P05771 1/20 0.40
CDK4 P11802 1/20 0.40
PRKCA P17252 1/20 0.40
PRKCH P24723 1/20 0.40
PRKCI P41743 1/20 0.40
PRKCE Q02156 1/20 0.40
KMT2A Q03164 1/20 0.40
PRKCQ Q04759 1/20 0.40
PRKCZ Q05513 1/20 0.40
PRKCD Q05655 1/20 0.40
PRKD1 Q15139 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TNIK Q9UKE5 1/20 0.40
GSK3A P49840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689717 0.82 MAOA (0.47) CHEK1CDK4
SCHEMBL8006987 0.70 TDP2 (0.48) WEE1CHEK1
SCHEMBL5829446 0.68 WEE1 (1.00) WEE1CHEK1ROCK2MEN1PRKD3
SCHEMBL31061050 0.68 WEE1 (1.00) WEE1CHEK1ROCK2MEN1PRKD3
SCHEMBL7912408 0.66 CYP1A2 (0.66) TDP1
SCHEMBL8694298 0.66 GNRHR (0.43)
SCHEMBL5828716 0.65 CHEK1 (1.00) WEE1CHEK1ROCK2MEN1PRKD3
SCHEMBL7905523 0.65 GAA (0.54) MEN1KMT2A
SCHEMBL8692753 0.65 GNRHR (0.42)
SCHEMBL8692748 0.65 GNRHR (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756507-A TREATING SEX HORMONE RELATED DISORDERS MERCK & CO., INC. (US) 1998-05-26 US disclosed