SCHEMBL8007796

SCHEMBL8007796

CC(Cn1ncc2ccc(S(C)(=O)=O)cc21)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.42
CA1 P00915 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
KMO O15229 4/20 0.41
GPR119 Q8TDV5 4/20 0.40
HTR2A P28223 4/20 0.39
HTR2C P28335 4/20 0.39
HTR2B P41595 3/20 0.39
HTR1A P08908 2/20 0.39
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
HTR1D P28221 1/20 0.39
HTR7 P34969 1/20 0.39
HTR4 Q13639 1/20 0.39
EEF2K O00418 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997838 0.84 KMO (0.43) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8007487 0.84 KMO (0.43) KMOHTR2AHTR2CHTR2BHTR1A
Fumaric Acid SCHEMBL8007684 0.72 HTR2A (0.56) KMOHTR2AHTR2CHTR2BHTR1A
Fumaric Acid SCHEMBL8009714 0.72 HTR2A (0.56) KMOHTR2AHTR2CHTR2BHTR1A
Fumaric Acid SCHEMBL8009708 0.72 HTR2A (0.56) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8007690 0.70 HTR2A (0.40) KMOGPR119HTR2AHTR2CHTR2B
SCHEMBL5636655 0.69 HTR2A (0.64) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL4946400 0.69 HTR2A (0.64) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL26988130 0.68 ITGA4 (0.36) CA2CA1CA4CA7CA9
SCHEMBL26989485 0.68 ITGA4 (0.36) CA2CA1CA4CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000017170-A2 N1-SUBSTITUTED BENZOPYRAZOLES AS INHIBITORS OF 5-HT2 RECEPTORS VERNALIS RESEARCH LIMITED (GB) 2000-03-30 WO disclosed