SCHEMBL8007698

SCHEMBL8007698

CCCn1c(-c2ccc(O)cc2)nc(-c2ccc(O)cc2)c1-c1ccc(O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.50
TEK Q02763 1/20 0.45
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
KDM4E B2RXH2 3/20 0.43
TSHR P16473 3/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GMNN O75496 1/20 0.43
USP2 O75604 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8011827 0.91 KDM4E (0.44) ESR1TEKKDM4ETSHRLMNA
SCHEMBL8011287 0.87 TEK (0.43) ESR1TEKKDM4ETSHRLMNA
SCHEMBL22219425 0.84 FAAH (0.49) TSHRTP53
SCHEMBL8008240 0.82 KDM4E (0.63) TEKKDM4ETSHRLMNANPSR1
SCHEMBL4422948 0.76 MLYCD (0.43) MAPK13MAPK12MAPK11MAPK14KDM4E
SCHEMBL18152846 0.75 TSHR (0.61) KDM4ETSHRHSD17B10TP53CYP1A2
SCHEMBL8797582 0.75 ALDH1A1 (0.53) KDM4ELMNANPSR1HSD17B10TP53
SCHEMBL7996428 0.74 KDM4E (0.53) TEKKDM4ETSHRLMNANPSR1
SCHEMBL27237042 0.74 FAAH (0.42) TP53MAPTADORA2BGAA
SCHEMBL8113557 0.74 FAAH (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000019994-A9 ESTROGEN RECEPTOR LIGANDS UNIV ILLINOIS (US) 2000-08-31 WO disclosed
WO-2000019994-A1 ESTROGEN RECEPTOR LIGANDS BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2000-04-13 WO disclosed