SCHEMBL8007487

SCHEMBL8007487

CC(Cn1ncc2ccc(I)cc21)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 6/20 0.43
HTR2A P28223 5/20 0.41
HTR2C P28335 5/20 0.41
HTR2B P41595 4/20 0.41
HTR1A P08908 2/20 0.41
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
HTR1D P28221 1/20 0.41
HTR7 P34969 1/20 0.41
HTR4 Q13639 1/20 0.41
PCSK9 Q8NBP7 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
TRPA1 O75762 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997838 1.00 KMO (0.43) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8007796 0.84 CA2 (0.42) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL24782853 0.78 KMO (0.45) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL26989485 0.75 ITGA4 (0.36) TRPA1MAPTITGA4ITGB7
SCHEMBL26988130 0.75 ITGA4 (0.36) TRPA1MAPTITGA4ITGB7
SCHEMBL26988251 0.75 ITGA4 (0.36) TRPA1MAPTITGA4ITGB7
SCHEMBL8007696 0.74 HTR2A (0.54) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL25702553 0.74 GABRG2 (0.46) KMOGABRG2GABRB3GABRA5GSK3B
SCHEMBL8007544 0.72 HTR2C (0.69) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8009907 0.72 HTR2C (0.69) KMOHTR2AHTR2CHTR2BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000017170-A2 N1-SUBSTITUTED BENZOPYRAZOLES AS INHIBITORS OF 5-HT2 RECEPTORS VERNALIS RESEARCH LIMITED (GB) 2000-03-30 WO disclosed