SCHEMBL8008273

SCHEMBL8008273

CCCCc1cc(-c2cccc(C=O)c2)ccc1COC(=O)c1cccc2nc(C)[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
KDM4E B2RXH2 2/20 0.32
BRS3 P32247 1/20 0.31
DHODH Q02127 1/20 0.30
EIF4A1 P60842 1/20 0.30
ALDH1A1 P00352 2/20 0.30
CYP3A4 P08684 2/20 0.30
TDP1 Q9NUW8 2/20 0.30
L3MBTL1 Q9Y468 2/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170666 0.71 TSHR (0.53) LMNAMAPTKDM4EALDH1A1L3MBTL1
SCHEMBL8357062 0.70 ALDH1A1 (0.36) LMNAMAPTKDM4EBRS3ALDH1A1
SCHEMBL12109510 0.64 KDM4E (0.46) LMNAMAPTKDM4EALDH1A1TDP1
SCHEMBL5970052 0.64 TSHR (0.55) LMNAKDM4EDHODHALDH1A1CYP3A4
SCHEMBL82573 0.63 TSHR (0.60) LMNAKDM4EALDH1A1CYP3A4TDP1
SCHEMBL8421782 0.63 ALDH1A1 (0.38) LMNAMAPTKDM4EALDH1A1CYP3A4
SCHEMBL6948237 0.62 TSHR (0.50) LMNAMAPTKDM4EALDH1A1TDP1
SCHEMBL9197306 0.62 RIPK1 (0.48) LMNAMAPTKDM4EALDH1A1L3MBTL1
SCHEMBL4713440 0.62 TSHR (0.52) LMNAKDM4EALDH1A1CYP3A4TDP1
SCHEMBL5734087 0.62 TRIM24 (0.50) MAPTTRIM24TRIM33ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100252-A SPECIFIED COMPOUNDS INCLUDING METHYL 2-BUTYL-1-((2'-(2-OXO-3H-1,2,3,5-OXATHIADIAZOL-4-YL)BIPHENYL) METHYL)-BENZIMIDAZOLE-7-CARBOXYLATE; USE TO TREAT CIRCULATORY DISEASES SUCH AS HYPERTENSIVE DISEASES AND HEART DISEASES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-08-08 US disclosed