SCHEMBL8008293

SCHEMBL8008293

COc1ccc(-n2nnc(C)n2)cc1CCCCCCc1nnc(C)o1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
ENPP2 Q13822 5/20 0.34
SPHK2 Q9NRA0 1/20 0.32
BRD9 Q9H8M2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 1/20 0.31
ABCB1 P08183 1/20 0.30
ABCG2 Q9UNQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009965 0.99 MTNR1A (0.36) MTNR1AMTNR1BENPP2SPHK2BRD9
SCHEMBL8008368 0.97 MTNR1A (0.36) MTNR1AMTNR1BENPP2BRD9ALDH1A1
SCHEMBL8014614 0.87 ENPP2 (0.32) MTNR1AMTNR1BENPP2
SCHEMBL8005853 0.82 ENPP2 (0.33) MTNR1AMTNR1BENPP2
SCHEMBL8010307 0.78 ENPP2 (0.34) MTNR1AMTNR1BENPP2BRD9ABCB1
SCHEMBL10260745 0.78 SPHK2 (0.32) SPHK2ABCB1ABCG2
SCHEMBL10260742 0.78 SPHK2 (0.32) SPHK2ABCB1ABCG2
SCHEMBL7999100 0.77 ALDH1A1 (0.39) ALDH1A1MAPTRAB9AGAA
SCHEMBL7999173 0.77 ALDH1A1 (0.39) ALDH1A1MAPTRAB9AGAA
SCHEMBL10292931 0.76 SPHK2 (0.33) SPHK2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed