SCHEMBL8010307

SCHEMBL8010307

COc1ccc(-n2nnc(C)n2)cc1/C=C/CCc1nnc(C)o1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 6/20 0.34
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
ABCB1 P08183 2/20 0.30
BRD9 Q9H8M2 2/20 0.30
ABCG2 Q9UNQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8015115 0.94 ENPP2 (0.34) ENPP2MTNR1AMTNR1B
SCHEMBL8005853 0.93 ENPP2 (0.33) ENPP2MTNR1AMTNR1B
SCHEMBL8009964 0.90 ENPP2 (0.34) ENPP2BRD9
SCHEMBL8000689 0.85 ENPP2 (0.32) ENPP2BRD9
SCHEMBL8009965 0.79 MTNR1A (0.36) ENPP2MTNR1AMTNR1BABCB1BRD9
SCHEMBL8008368 0.79 MTNR1A (0.36) ENPP2MTNR1AMTNR1BABCB1BRD9
SCHEMBL8005747 0.78 ALDH1A1 (0.37)
SCHEMBL8008293 0.78 MTNR1A (0.35) ENPP2MTNR1AMTNR1BABCB1BRD9
SCHEMBL8005781 0.78 ALDH1A1 (0.37)
SCHEMBL10293193 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed