SCHEMBL8009944

SCHEMBL8009944

COc1ccnc(C[C@@H](N)C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.49
NOS1 P29475 2/20 0.49
NOS2 P35228 2/20 0.49
CYP1A2 P05177 1/20 0.47
TPH1 P17752 3/20 0.43
LNPEP Q9UIQ6 3/20 0.43
CCR1 P32246 1/20 0.42
CCR5 P51681 1/20 0.42
CCR8 P51685 1/20 0.42
SLC7A5 Q01650 2/20 0.42
PLAU P00749 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GRIK1 P39086 1/20 0.41
GRIK2 Q13002 1/20 0.41
LDHA P00338 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4871525 0.84 NOS3 (0.50) NOS3NOS1NOS2CYP1A2LNPEP
SCHEMBL5566353 0.79 HSD17B10 (0.50) NOS3NOS1NOS2CYP1A2SLC7A5
SCHEMBL31369944 0.79 TPH1 (0.54) TPH1CCR1CCR5CCR8SLC7A5
SCHEMBL8000728 0.78 CYP1A2 (0.51) CYP1A2SLC7A5HSD17B10LMNA
SCHEMBL22775125 0.78 CYP1A2 (0.51) CYP1A2SLC7A5HSD17B10LMNA
SCHEMBL24248055 0.77 HSD17B10 (0.51) CYP1A2SLC7A5HSD17B10
SCHEMBL15495937 0.77 HSD17B10 (0.51) CYP1A2SLC7A5HSD17B10LMNA
SCHEMBL18995811 0.77 HSD17B10 (0.51) CYP1A2SLC7A5HSD17B10
SCHEMBL20278960 0.77 NOS2 (0.49) NOS3NOS1NOS2CCR1CCR5
SCHEMBL15743142 0.76 NOS3 (0.56) NOS3NOS1NOS2CYP1A2CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850316-A4 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIV HAWAII (US) 2000-08-23 EP disclosed
EP-0850316-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1998-07-01 EP disclosed
WO-1997008334-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1997-03-06 WO disclosed