SCHEMBL8010408

SCHEMBL8010408

Cc1c(S(Cl)(Cl)CF)c(C#N)c(Cl)n1-c1c(Cl)cc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.38
CYP3A4 P08684 4/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
HIF1A Q16665 1/20 0.38
TXNRD1 Q16881 1/20 0.38
TXNRD3 Q86VQ6 1/20 0.38
TXNRD2 Q9NNW7 1/20 0.38
MAPK1 P28482 6/20 0.37
LMNA P02545 4/20 0.37
GABRB3 P28472 3/20 0.34
GABRA2 P47869 3/20 0.34
GABRB2 P47870 3/20 0.34
GABRP O00591 2/20 0.34
GABRD O14764 2/20 0.34
GABRA1 P14867 2/20 0.34
GABRB1 P18505 2/20 0.34
GABRG2 P18507 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026720 0.88 GABRB3 (0.40) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL8446583 0.81 GABRB3 (0.41) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL7812035 0.79 TDP1 (0.39) TDP1CYP3A4TSHRALDH1A1HPGD
SCHEMBL9028146 0.76 GABRB3 (0.38) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL9028687 0.75 GABRP (0.37) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL8822800 0.75 GABRB3 (0.45) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL7825839 0.73 TDP1 (0.41) TDP1CYP3A4TSHRALDH1A1HPGD
SCHEMBL8446016 0.70 GABRA2 (0.41) CYP3A4LMNAGABRB3GABRA2GABRB2
SCHEMBL3033497 0.69 ALDH1A1 (0.59) TDP1CYP3A4TSHRALDH1A1HPGD
SCHEMBL8822967 0.68 GABRA2 (0.40) CYP3A4LMNAGABRB3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0738713-B1 Process for the preparation of pesticidal 1-(chloroaryl)heterocyclic compounds RHONE POULENC AGROCHIMIE (FR) 2000-02-09 EP disclosed
US-5726324-A 1-(nitroaryl)pyrrole intermediates to pesticidal 1-(haloaryl)pyrroles RHONE-POULENC INC. (US) 1998-03-10 US disclosed
US-5631381-A Process for the preparation of pesticidal 1-(haloaryl) heterocyclic compounds RHONE-POULENC INC. (US) 1997-05-20 US disclosed
EP-0738713-A1 Process for the preparation of pesticidal 1-(haloaryl)heterocyclic compounds RHONE-POULENC AGROCHIMIE (FR) 1996-10-23 EP disclosed