SCHEMBL8010665

SCHEMBL8010665

CCc1nc(-c2cc[c]cc2)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
DDAH1 O94760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457222 0.81 SMN1; SMN2 (0.56) SMN1; SMN2ADORA3ADORA2AADORA1DDAH1
SCHEMBL27909694 0.80 RAD51 (0.42) SMN1; SMN2ADORA3ADORA1
SCHEMBL14039561 0.80 METAP2 (0.47) SMN1; SMN2
SCHEMBL948854 0.80 GSK3B (0.44) SMN1; SMN2
SCHEMBL19405233 0.79 ALDH1A1 (0.39) SMN1; SMN2ADORA3ADORA2AADORA1
SCHEMBL8012285 0.79 TLR8 (0.39) SMN1; SMN2ADORA3ADORA2AADORA1
SCHEMBL28079633 0.79 NPC1 (0.42) SMN1; SMN2ADORA2AADORA1
SCHEMBL4415849 0.76 GSK3B (0.33)
SCHEMBL17599659 0.75 HEXA (0.42) ADORA3
SCHEMBL11208038 0.75 SMN1; SMN2 (0.39) SMN1; SMN2ADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US claimed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO claimed
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed