SCHEMBL8012736

SCHEMBL8012736

CN1CCc2sccc2C1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 3/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35
GID4 Q8IVV7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021988 0.77 KMT2A (0.51) HHATKMT2ADRD2DRD3DRD1
SCHEMBL22044650 0.77 KMT2A (0.51) HHATKMT2ADRD2DRD3DRD1
SCHEMBL8026946 0.72 DRD2 (0.42) HHATKMT2ADRD2DRD3DRD1
SCHEMBL8025796 0.70 PRCP (0.56) DRD2DRD1DRD4DRD5
SCHEMBL8030400 0.67 MEN1 (0.42) KMT2ADRD2DRD3DRD1DRD4
SCHEMBL8030423 0.67 SRD5A1 (0.43) DRD2DRD1DRD4
SCHEMBL8032022 0.67 HTR2A (0.43) DRD2
SCHEMBL4751918 0.67 DRD2 (0.42) HHATKMT2ADRD2DRD3DRD1
SCHEMBL22679819 0.66 KMT2A (0.48) HHATKMT2ADRD2DRD3DRD1
SCHEMBL2836823 0.66 DRD1 (0.41) HHATKMT2ADRD2DRD3DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095253-A1 6-HALO-PYRAZOLO[1, 5-A]PYRIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR (MGLUR) MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2009-08-06 WO disclosed