SCHEMBL8014129

SCHEMBL8014129

COc1cc(C(C)Nc2ncnc(C(C)F)c2Cl)ccc1OC(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.43
SOS1 Q07889 2/20 0.43
KRAS P01116 1/20 0.43
HDAC3 O15379 4/20 0.37
HDAC4 P56524 4/20 0.37
HDAC1 Q13547 4/20 0.37
HDAC7 Q8WUI4 4/20 0.37
HDAC2 Q92769 4/20 0.37
HDAC10 Q969S8 4/20 0.37
HDAC11 Q96DB2 4/20 0.37
HDAC8 Q9BY41 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
HDAC9 Q9UKV0 4/20 0.37
HDAC5 Q9UQL6 4/20 0.37
ERBB2 P04626 2/20 0.37
P2RX3 P56373 1/20 0.37
PDE5A O76074 1/20 0.37
RPS6KB1 P23443 1/20 0.36
KDR P35968 1/20 0.36
RET P07949 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025127 0.93 EGFR (0.46) EGFRSOS1KRASHDAC3HDAC4
SCHEMBL8024922 0.89 EGFR (0.42) EGFRSOS1KRASP2RX3PDE5A
SCHEMBL9728955 0.83 EGFR (0.43) EGFRSOS1KRASP2RX3
SCHEMBL8024509 0.81 EGFR (0.40) EGFRSOS1KRAS
SCHEMBL9729028 0.80 EGFR (0.41) EGFRSOS1KRASERBB2
SCHEMBL8024930 0.80 EGFR (0.48) EGFRSOS1KRASP2RX3RPS6KB1
SCHEMBL8025390 0.80 EGFR (0.42) EGFRSOS1KRASRPS6KB1
SCHEMBL8014462 0.77 CYP2D6 (0.49) EGFRSOS1KRASCA1CA2
SCHEMBL8026893 0.77 EGFR (0.37) EGFRSOS1KRASRPS6KB1
SCHEMBL16997376 0.76 EGFR (0.41) EGFRSOS1KRASP2RX3RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543402-B1 Aralkylaminopyrimidine derivative, method for preparing the same and composition for controlling noxious organisms UBE INDUSTRIES (JP) 2000-03-01 EP claimed
US-5280025-A Aralkylaminopyrimidine derivative, and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1994-01-18 US claimed
EP-0543402-A1 Aralkylaminopyrimidine derivative, method for preparing the same and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1993-05-26 EP claimed