SCHEMBL8014258

SCHEMBL8014258

CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COC(c1ccccc1)(c1ccc(OC)cc1)c1ccc(OC)cc1)OC(=O)CCCCCCC/C=C\CCCCCCCC

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 3/20 0.54
PRKCE Q02156 2/20 0.54
PRKCQ Q04759 2/20 0.54
PRKCD Q05655 2/20 0.54
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
LPAR1 Q92633 2/20 0.48
SELP P16109 1/20 0.47
DAGLA Q9Y4D2 1/20 0.46
ENPP2 Q13822 2/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LPAR3 Q9UBY5 1/20 0.46
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL978433 0.92 PRKCA (0.59) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL975774 0.92 PRKCA (0.59) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL974889 0.92 PRKCA (0.59) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL4981050 0.88 ENPP2 (0.60) PRKCAPRKCEPRKCQPRKCDLPAR1
SCHEMBL4981054 0.88 ENPP2 (0.60) PRKCAPRKCEPRKCQPRKCDLPAR1
SCHEMBL9453916 0.88 PRKCA (0.53) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL18660350 0.86 ALDH1A1 (0.44) ALDH1A1DAGLACNR1
SCHEMBL18660352 0.84 ALDH1A1 (0.42) ALDH1A1DAGLACNR1
SCHEMBL18660354 0.84 ALDH1A1 (0.42) ALDH1A1DAGLACNR1
SCHEMBL6346855 0.81 DGKA (0.60) PRKCEPRKCQPRKCDLPAR1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685234-B1 DRUG COMPOSITION CONTAINING NUCLEIC ACID COPOLYMER NIPPON SHINYAKU CO LTD (JP) 2000-05-10 EP disclosed
US-6020317-A Glycerol derivative, device and pharmaceutical composition NIPPON SHINYAKU CO. LTD. (JP) 2000-02-01 US disclosed
EP-0685457-B1 GLYCEROL DERIVATIVE, DEVICE AND PHARMACEUTICAL COMPOSITION NIPPON SHINYAKU CO LTD (JP) 1999-12-15 EP disclosed
US-5705188-A LIPID MIXTURE, ANTITUMOR AGENTS NIPPON SHINYAKU COMPANY, LTD. (JP) 1998-01-06 US disclosed
EP-0685457-A1 GLYCEROL DERIVATIVE, DEVICE AND PHARMACEUTICAL COMPOSITION NIPPON SHINYAKU COMPANY, LIMITED (JP) 1995-12-06 EP disclosed
EP-0685234-A1 DRUG COMPOSITION CONTAINING NUCLEIC ACID COPOLYMER NIPPON SHINYAKU COMPANY, LIMITED (JP) 1995-12-06 EP disclosed
US-5248618-A METHODS FOR GENERATING LIGHT WITH CHEMILUMINESCENT DIOXETANES ACTIVATED BY ANCHIMERIC ASSISTED CLEAVAGE LIFE TECHNOLOGIES, INC. (US) 1993-09-28 US disclosed
WO-1992021778-A1 ASSAYS EMPLOYING ANCHIMERIC ASSISTANCE CLEAVAGE LIFE TECHNOLOGIES, INC. (US) 1992-12-10 WO disclosed