SCHEMBL8014589

SCHEMBL8014589

CC(F)c1ncnc(NCC2(c3ccc(Cl)cc3)CC2)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.41
SLC6A3 Q01959 6/20 0.41
SLC6A2 P23975 3/20 0.41
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36
P2RX3 P56373 1/20 0.35
F2 P00734 1/20 0.35
CNR1 P21554 2/20 0.33
AKT2 P31751 1/20 0.33
GSK3B P49841 1/20 0.33
P2RX7 Q99572 2/20 0.32
MAPT P10636 1/20 0.32
CHRM2 P08172 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
HTR2A P28223 1/20 0.32
OPRK1 P41145 1/20 0.32
HTR2B P41595 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024811 0.89 SLC6A4 (0.34) SLC6A4SLC6A3SLC6A2CTSDBACE1
SCHEMBL8014400 0.88 SLC6A4 (0.32) SLC6A4SLC6A3
SCHEMBL8014567 0.87 P2RX7 (0.40) SLC6A4SLC6A3P2RX7EGFR
SCHEMBL9329582 0.84 SLC6A4 (0.50) SLC6A4SLC6A3SLC6A2
SCHEMBL8024318 0.79 EGFR (0.51) CNR1MAPTEGFRACACBCNR2
SCHEMBL8024821 0.76 CLK4 (0.32)
SCHEMBL8026802 0.71 CDK1 (0.50) EGFR
SCHEMBL8025185 0.70 PRMT1 (0.48) P2RX7MAPTEGFRTP53
SCHEMBL8024781 0.68 HTT (0.55) P2RX7MAPTEGFRTP53
SCHEMBL8014586 0.68 SLC6A4 (0.36) SLC6A4SLC6A3SLC6A2MAPTCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543402-B1 Aralkylaminopyrimidine derivative, method for preparing the same and composition for controlling noxious organisms UBE INDUSTRIES (JP) 2000-03-01 EP claimed
US-5280025-A Aralkylaminopyrimidine derivative, and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1994-01-18 US claimed
EP-0543402-A1 Aralkylaminopyrimidine derivative, method for preparing the same and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1993-05-26 EP claimed
EP-0543402-B1 Aralkylaminopyrimidine derivative, method for preparing the same and composition for controlling noxious organisms UBE INDUSTRIES (JP) 2000-03-01 EP disclosed
US-5280025-A Aralkylaminopyrimidine derivative, and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1994-01-18 US disclosed
EP-0543402-A1 Aralkylaminopyrimidine derivative, method for preparing the same and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1993-05-26 EP disclosed