SCHEMBL8015385

SCHEMBL8015385

CCOc1nc(C)cc2nc(S(=O)(=O)Cl)nn12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GLA P06280 1/20 0.33
MAPT P10636 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PKM P14618 3/20 0.32
MAPK1 P28482 2/20 0.32
HSD17B10 Q99714 1/20 0.32
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
AHR P35869 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559900 0.86 PDE4D (0.33) MAPTSMN1; SMN2
SCHEMBL6998020 0.85 GNRHR (0.32) MAPTKDM4EALDH1A1POLBHPGD
SCHEMBL8025547 0.84 KDM4E (0.35) MEN1KMT2AMAPTSMN1; SMN2PKM
SCHEMBL9642094 0.79 JAK1 (0.35) PKM
SCHEMBL10749665 0.77 PDE10A (0.36) MAPTSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL10490295 0.77 MEN1 (0.42) L3MBTL1MEN1KMT2AGLAMAPT
SCHEMBL8881335 0.76 TSHR (0.37) MAPTKDM4EALDH1A1POLBNPSR1
SCHEMBL8798465 0.75 NPC1 (0.32) MEN1KMT2APKMHSD17B10KDM4E
SCHEMBL8882800 0.74 TSHR (0.32)
SCHEMBL9642675 0.74 ADORA3 (0.37) MAPTMAPK1HSD17B10ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888297-B1 N-ARYLSULFILIMINE COMPOUNDS AND THEIR USE AS CATALYSTS IN THE PREPARATION OF N-ARYLARYLSULFONAMIDE COMPOUNDS DOW AGROSCIENCES LLC (US) 2000-08-30 EP claimed
US-5973148-A N-arylsulfilimine compounds and their use as catalysts in the preparation of N-arylarylsulfonamide compounds DOW AGROSCIENCES LLC (US) 1999-10-26 US claimed
US-6162915-A Process for heterocyclic sulfonyl chloride compounds DOW AGROSCIENCES LLC (US) 2000-12-19 US disclosed
US-6114580-A N-arylsulfilimine compounds and their use as catalysts in the preparation of N-arylarylsulfonamide compounds DOW AGROSCIENCES LLC (US) 2000-09-05 US disclosed
EP-0888297-B1 N-ARYLSULFILIMINE COMPOUNDS AND THEIR USE AS CATALYSTS IN THE PREPARATION OF N-ARYLARYLSULFONAMIDE COMPOUNDS DOW AGROSCIENCES LLC (US) 2000-08-30 EP disclosed
US-5973148-A N-arylsulfilimine compounds and their use as catalysts in the preparation of N-arylarylsulfonamide compounds DOW AGROSCIENCES LLC (US) 1999-10-26 US disclosed
EP-0922047-A1 PROCESS FOR HETEROCYCLIC SULFONYL CHLORIDE COMPOUNDS Dow AgroSciences LLC (US) 1999-06-16 EP disclosed
WO-1999000392-A1 PROCESS FOR HETEROCYCLIC SULFONYL CHLORIDE COMPOUNDS DOW AGROSCIENCES LLC (US) 1999-01-07 WO disclosed
EP-0537611-B1 Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOW AGROSCIENCES LLC (US) 1998-08-12 EP disclosed
EP-0343752-B1 Alkoxy-1,2,4-triazolo (1,5-c) pyrimidine-2-sulfonamides, process for their preparation and intermediates DOWELANCO (US) 1993-12-01 EP disclosed
EP-0537611-A1 Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOWELANCO (US) 1993-04-21 EP disclosed
US-5177206-A Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOWELANCO (US) 1993-01-05 US disclosed
US-5163995-A For use with grassy crops and soybeans DOWELANCO (US) 1992-11-17 US disclosed
WO-1989011782-A1 ALKOXY-1,2,4-TRIAZOLO[1,5-c]PYRIMIDINE-2-SULFONAMIDES, PROCESS FOR THEIR PREPARATION AND INTERMEDIATES THE DOW CHEMICAL COMPANY (US) 1989-12-14 WO disclosed
EP-0343752-A1 Alkoxy-1,2,4-triazolo (1,5-c) pyrimidine-2-sulfonamides, process for their preparation and intermediates DowElanco (US) 1989-11-29 EP disclosed