SCHEMBL8015840

SCHEMBL8015840

CN(Cc1ccccc1)c1nc2c(S(=O)(=O)c3ccc(F)cc3)nnn2c2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.67
HTR6 P50406 11/20 0.64
RXFP1 Q9HBX9 3/20 0.63
THRB P10828 1/20 0.54
KDM4E B2RXH2 3/20 0.50
HPGD P15428 2/20 0.50
ALDH1A1 P00352 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8019490 0.93 HTR6 (0.72) TP53HTR6RXFP1THRBKDM4E
SCHEMBL8027148 0.90 RXFP1 (0.65) TP53HTR6RXFP1THRBKDM4E
SCHEMBL8018281 0.87 HPGD (0.53) TP53HTR6RXFP1THRBKDM4E
SCHEMBL8030780 0.85 HTR6 (0.65) TP53HTR6RXFP1THRBPOLB
SCHEMBL8019551 0.84 HTR6 (0.75) TP53HTR6RXFP1THRBKDM4E
SCHEMBL8018278 0.80 HPGD (0.60) TP53HTR6RXFP1THRBKDM4E
SCHEMBL8029679 0.80 TP53 (1.00) TP53HTR6RXFP1THRBSMN1; SMN2
SCHEMBL8028973 0.78 HTR6 (0.73) TP53HTR6RXFP1THRB
SCHEMBL8029076 0.78 HTR6 (1.00) TP53HTR6RXFP1
SCHEMBL8029045 0.77 KDM4E (0.61) TP53HTR6RXFP1THRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed