SCHEMBL8019490

SCHEMBL8019490

CN(Cc1ccccc1)c1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 11/20 0.72
TP53 P04637 1/20 0.69
RXFP1 Q9HBX9 3/20 0.66
THRB P10828 1/20 0.56
KDM4E B2RXH2 3/20 0.56
ALDH1A1 P00352 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
POLB P06746 1/20 0.56
HPGD P15428 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8015840 0.93 TP53 (0.67) HTR6TP53RXFP1THRBKDM4E
SCHEMBL8027148 0.91 RXFP1 (0.65) HTR6TP53RXFP1THRBKDM4E
SCHEMBL8019551 0.91 HTR6 (0.75) HTR6TP53RXFP1THRBKDM4E
SCHEMBL8018278 0.87 HPGD (0.60) HTR6TP53RXFP1THRBKDM4E
SCHEMBL8029076 0.84 HTR6 (1.00) HTR6TP53RXFP1
SCHEMBL8028973 0.84 HTR6 (0.73) HTR6TP53RXFP1THRB
SCHEMBL8029045 0.84 KDM4E (0.61) HTR6TP53RXFP1THRBKDM4E
SCHEMBL8029679 0.82 TP53 (1.00) HTR6TP53RXFP1THRB
SCHEMBL8028235 0.79 HTR6 (0.89) HTR6RXFP1
SCHEMBL8018281 0.78 HPGD (0.53) HTR6TP53RXFP1THRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed