SCHEMBL8018281

SCHEMBL8018281

CN(C)c1nc2c(S(=O)(=O)c3ccc(F)cc3)nnn2c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 7/20 0.53
ALDH1A1 P00352 7/20 0.53
KDM4E B2RXH2 5/20 0.53
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
KMT2A Q03164 3/20 0.52
GAA P10253 2/20 0.52
RXFP1 Q9HBX9 4/20 0.52
NPSR1 Q6W5P4 2/20 0.52
MAPT P10636 3/20 0.51
RECQL P46063 1/20 0.51
MEN1 O00255 1/20 0.51
POLB P06746 1/20 0.50
TP53 P04637 1/20 0.49
HTR6 P50406 4/20 0.48
THRB P10828 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8018278 0.91 HPGD (0.60) HPGDALDH1A1KDM4ECRHBPCRHR2
SCHEMBL8019463 0.88 HPGD (0.53) HPGDALDH1A1KDM4ECRHBPCRHR2
SCHEMBL8015840 0.87 TP53 (0.67) HPGDALDH1A1KDM4ERXFP1NPSR1
SCHEMBL8019456 0.82 KDM4E (0.64) HPGDALDH1A1KDM4ECRHBPCRHR2
SCHEMBL8019460 0.82 HTR6 (0.60) HPGDALDH1A1KDM4EGAARXFP1
SCHEMBL8028247 0.81 HTR6 (0.48) RXFP1MAPTPOLBHTR6
SCHEMBL8029045 0.79 KDM4E (0.61) HPGDALDH1A1KDM4ECRHBPCRHR2
SCHEMBL8019490 0.78 HTR6 (0.72) HPGDALDH1A1KDM4ERXFP1NPSR1
SCHEMBL10123316 0.76 THRB (0.63) HPGDALDH1A1KDM4EGAARXFP1
SCHEMBL8030043 0.75 HTR6 (0.50) HPGDALDH1A1KDM4ECRHBPCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed