SCHEMBL8017016

SCHEMBL8017016

NC(=O)CCc1coc2ccc(O)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.54
HTR1D P28221 2/20 0.54
HTR2C P28335 2/20 0.54
MTNR1B P49286 2/20 0.47
SIRT1 Q96EB6 4/20 0.46
ALDH1A1 P00352 2/20 0.44
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
NPC1 O15118 2/20 0.43
CASP3 P42574 2/20 0.43
SENP7 Q9BQF6 2/20 0.43
SENP6 Q9GZR1 2/20 0.43
SENP8 Q96LD8 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 1/20 0.43
NFKB1 P19838 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8690961 0.88 PIM1 (0.53) HTR1AHTR1DHTR2CALDH1A1TSHR
SCHEMBL8690168 0.86 HTR1A (0.48) HTR1AHTR1DHTR2CMTNR1BSIRT1
SCHEMBL7019210 0.81 MTNR1A (0.49) HTR1AHTR1DHTR2CMTNR1BSIRT1
SCHEMBL8695023 0.80 MTNR1A (0.65) HTR2CMTNR1BALDH1A1TSHRNPC1
SCHEMBL11365468 0.80 MAOB (0.51) HTR1AHTR1DHTR2CMAOB
SCHEMBL7014521 0.78 HTR1A (0.47) HTR1AHTR1DHTR2CMTNR1BSIRT1
SCHEMBL2269511 0.78 MTNR1A (0.51) HTR1AHTR1DHTR2CMTNR1BSIRT1
SCHEMBL2267233 0.77 NPC1 (0.49) SIRT1ALDH1A1TSHRNPSR1MAPT
SCHEMBL24938760 0.76 ALOX15 (0.59) SIRT1ALDH1A1TSHRNPSR1MAPT
SCHEMBL5340289 0.76 MTNR1A (0.48) HTR1AHTR1DHTR2CMTNR1BSIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745584-B1 Arylalkyl(thio) carboxamides compounds with affinity for melatonine receptors, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-01-05 EP disclosed
US-5721276-A TREATING DISORDERS OF MELATONINERGIC SYSTEM ADIR ET COMPAGNIE (FR) 1998-02-24 US disclosed
EP-0745584-A1 Arylalkyl(thio) carboxamides compounds with affinity for melatonine receptors, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-12-04 EP disclosed