SCHEMBL8017172

SCHEMBL8017172

O=C(Cl)c1ccccc1OBr

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
ALOX15 P16050 2/20 0.48
HTT P42858 3/20 0.40
KMT2A Q03164 3/20 0.40
CTSD P07339 1/20 0.40
TP53 P04637 1/20 0.39
KDM4E B2RXH2 4/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 4/20 0.38
ESR1 P03372 2/20 0.38
TSHR P16473 2/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
HMGB1 P09429 1/20 0.38
GGT1 P19440 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
BLM P54132 1/20 0.38
NAPRT Q6XQN6 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3357655 0.82 ALDH1A1 (0.52) ALDH1A1ALOX15HTTKMT2ACTSD
SCHEMBL16669782 0.80 ALDH1A1 (0.50) ALDH1A1ALOX15HTTKMT2ACTSD
SCHEMBL5427931 0.80 KDM4E (0.59) ALDH1A1ALOX15HTTKMT2ATP53
SCHEMBL431 0.78 CTSD (0.63) ALDH1A1HTTCTSDTP53HPGD
SCHEMBL1996334 0.78 CTNNB1 (0.60) ALDH1A1HTTKMT2AKDM4EHPGD
SCHEMBL29392137 0.78 CTSD (0.63) ALDH1A1HTTCTSDTP53HPGD
SCHEMBL7910478 0.78 ALDH1A1 (0.44) ALDH1A1ALOX15HTTKMT2ACTSD
SCHEMBL27972601 0.78 ALDH1A1 (0.44) ALDH1A1ALOX15HTTKMT2ACTSD
Water SCHEMBL29682837 0.77 KDM4E (0.55) ALDH1A1ALOX15HTTKMT2ATP53
SCHEMBL28432969 0.77 KMT2A (0.63) ALDH1A1ALOX15HTTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885199-A4 KAPPA AGONIST COMPOUNDS AND PHARMACEUTICAL FORMULATIONS THEREOF ADOLOR CORP (US) 2000-11-29 EP disclosed
EP-0885199-A1 KAPPA AGONIST COMPOUNDS AND PHARMACEUTICAL FORMULATIONS THEREOF Adolor Corporation (US) 1998-12-23 EP disclosed
WO-1997032857-A1 KAPPA AGONIST COMPOUNDS AND PHARMACEUTICAL FORMULATIONS THEREOF ADOLOR CORPORATION (US) 1997-09-12 WO disclosed