SCHEMBL8017607

SCHEMBL8017607

C[C](c1ccccc1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.44
CES1 P23141 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MAPT P10636 2/20 0.41
LMNA P02545 2/20 0.41
XBP1 P17861 1/20 0.41
ATM Q13315 1/20 0.41
ELANE P08246 2/20 0.40
ALDH1A1 P00352 3/20 0.39
HTT P42858 2/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
TSHR P16473 3/20 0.39
DAO P14920 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
HTR2A P28223 2/20 0.38
ESR1 P03372 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1518530 0.77 PTGS2 (0.44) SMN1; SMN2MAPTLMNAALDH1A1HPGD
SCHEMBL4578842 0.75 LMNA (0.41) CES2CES1SMN1; SMN2MAPTLMNA
SCHEMBL28158669 0.74 SMN1; SMN2 (0.43) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL3244408 0.74 NPSR1 (0.43) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL7370238 0.74 SMN1; SMN2 (0.43) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL13651331 0.74 ESR1 (0.45) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL6535707 0.74 ESR1 (0.45) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL28287732 0.74 GAA (0.42) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL19624236 0.74 ESR1 (0.45) CES2CES1SMN1; SMN2NPSR1MAPT
SCHEMBL5013786 0.74 TDP1 (0.54) CES2CES1LMNAATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016087593-A1 NOVEL FUNGICIDAL QUINOLINYLAMIDINES SYNGENTA PARTICIPATIONS AG (CH) 2016-06-09 WO disclosed
US-6103732-A ENDOTHELIN RECEPTOR INHIBITORS; HYPOTENSIVE AGENTS, CARDIOTONIC AGENTS; ACUTE MYOCARDIAL INFARCT, PULMONARY HYPERTENSION, RAYNAUD'S SYNDROME, ATHEROSCLEROSIS; ASTHMA; CARDIOVASCULAR DISORDERS BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed
US-6051569-A 1'S, 5R, 6R-carbapenem derivatives and antimicrobial agents comprising the same SUNTORY LIMITED (JP) 2000-04-18 US disclosed
EP-0826687-A1 Carbapenem derivatives and antimicrobial agents comprising the same SUNTORY LIMITED (JP) 1998-03-04 EP disclosed
EP-0414200-B1 Salts of optically active 4-hydroxy-8-(3-lower alkoxy-4-phenylsulfinylphenyl)pyrazolo [1,5-a]-1,3,5-triazines and a process for production thereof OTSUKA PHARMA CO LTD (JP) 1995-08-02 EP disclosed
CN-1028528-C Salts of optically active 4-hydroxy-8-(3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a]-1,3,5-triazines OTSUKA PHARMA CO LTD (JP) 1995-05-24 CN disclosed
EP-0572547-A1 SUBSTITUTED $g(a)-AMINOALDEHYDES AND DERIVATIVES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-12-08 EP disclosed
US-5180799-A Organolithium-Organoaluminum Catalyst IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-01-19 US disclosed
US-5137887-A Xanthine oxidase inhibitors, antipodagric agents OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1992-08-11 US disclosed
EP-0434316-A1 Processes ZENECA LIMITED (GB) 1991-06-26 EP disclosed
CN-1049664-A Optically active 4-hydroxyl-8-(3-low-alkoxy-4-phenyl sulfinyl phenyl) pyrazolo [1,5-α]-1,3,5-triazines salt and method for making thereof OTSUKA PHARMA CO LTD (JP) 1991-03-06 CN disclosed
EP-0414200-A2 Salts of optically active 4-hydroxy-8-(3-lower alkoxy-4-phenylsulfinylphenyl)pyrazolo [1,5-a]-1,3,5-triazines and a process for production thereof OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1991-02-27 EP disclosed
US-4963582-A ANTHELMINTICS, ACARICIDES, INSECTICIDES SANKYO COMPANY LIMITED (JP) 1990-10-16 US disclosed