SCHEMBL8019079

SCHEMBL8019079

O=S(=O)(c1ccccc1)c1nnn2c1ncc1ccccc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
HPGD P15428 5/20 0.51
HTR6 P50406 11/20 0.50
ALDH1A1 P00352 5/20 0.50
RXFP1 Q9HBX9 4/20 0.50
NPSR1 Q6W5P4 2/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 3/20 0.48
RECQL P46063 1/20 0.48
GAA P10253 1/20 0.47
TP53 P04637 2/20 0.47
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8030043 0.90 HTR6 (0.50) KDM4EHPGDHTR6ALDH1A1RXFP1
SCHEMBL8021669 0.86 HPGD (0.45) KDM4EHPGDHTR6ALDH1A1RXFP1
SCHEMBL8019100 0.86 HTR6 (0.57) HTR6RXFP1MAPTGAATP53
SCHEMBL8018264 0.79 HTR6 (0.52) HTR6RXFP1MAPTTP53
SCHEMBL8018278 0.73 HPGD (0.60) KDM4EHPGDHTR6ALDH1A1RXFP1
SCHEMBL8021786 0.73 KDM4E (0.72) KDM4EHPGDHTR6ALDH1A1RXFP1
SCHEMBL14349689 0.71 KDM4E (0.40) KDM4EHPGDALDH1A1RXFP1NPSR1
SCHEMBL10666827 0.71 KDM4E (0.40) KDM4EHPGDALDH1A1RXFP1NPSR1
SCHEMBL10668591 0.71 KDM4E (0.44) KDM4EHPGDALDH1A1RXFP1NPSR1
SCHEMBL8028196 0.71 HPGD (0.84) KDM4EHPGDHTR6ALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed