SCHEMBL8021669

SCHEMBL8021669

O=S(=O)(c1cccc(F)c1)c1nnn2c1ncc1ccccc12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.45
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 5/20 0.45
MAPT P10636 5/20 0.45
RECQL P46063 1/20 0.45
TP53 P04637 2/20 0.44
RXFP1 Q9HBX9 4/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HTR6 P50406 9/20 0.43
GAA P10253 2/20 0.42
KMT2A Q03164 1/20 0.42
THRB P10828 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8030043 0.87 HTR6 (0.50) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8019079 0.86 KDM4E (0.51) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8026985 0.81 HTR6 (0.46) MAPTRXFP1HTR6GAA
SCHEMBL8019463 0.77 HPGD (0.53) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8021789 0.77 KDM4E (0.64) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8027148 0.72 RXFP1 (0.65) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8018264 0.68 HTR6 (0.52) MAPTTP53RXFP1HTR6
SCHEMBL8028243 0.68 HTR6 (0.59) MAPTTP53RXFP1HTR6GAA
SCHEMBL8028518 0.66 HTR6 (0.55) MAPTTP53RXFP1HTR6GAA
SCHEMBL8018356 0.66 HTR6 (0.48) MAPTRXFP1HTR6GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed