SCHEMBL8019337

SCHEMBL8019337

O=C1C(=O)N(Cc2ccccc2)c2ccc([N+](=O)[O-])cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 1.00
CASP7 P55210 4/20 1.00
CASP6 P55212 4/20 1.00
CASP1 P29466 2/20 1.00
CASP4 P49662 2/20 1.00
CASP9 P55211 2/20 1.00
CASP8 Q14790 1/20 1.00
ALDH1A1 P00352 4/20 0.70
HPGD P15428 1/20 0.70
HTT P42858 1/20 0.70
CA12 O43570 2/20 0.66
CA1 P00915 2/20 0.66
CA2 P00918 2/20 0.66
CA9 Q16790 2/20 0.66
ALDH2 P05091 3/20 0.64
ALDH3A1 P30838 3/20 0.64
KDM1A O60341 1/20 0.62
CHRM1 P11229 1/20 0.60
CES1 P23141 1/20 0.60
APP P05067 4/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27881879 0.89 CASP3 (0.81) CASP3CASP7CASP6CASP1CASP4
SCHEMBL8019897 0.88 CASP3 (0.79) CASP3CASP7CASP6CASP1CASP4
SCHEMBL1217303 0.87 CASP3 (0.77) CASP3CASP7CASP6CASP1CASP4
SCHEMBL9094786 0.85 CASP1 (0.73) CASP3CASP7CASP6CASP1CASP4
SCHEMBL28026201 0.85 CASP1 (0.73) CASP3CASP7CASP6CASP1CASP4
SCHEMBL28365949 0.84 CASP1 (0.72) CASP3CASP7CASP6CASP1CASP4
SCHEMBL13627910 0.84 CASP1 (0.72) CASP3CASP7CASP6CASP1CASP4
SCHEMBL18954667 0.83 ALDH1A1 (0.74) CASP3CASP7CASP6CASP1CASP4
SCHEMBL18954527 0.83 CASP1 (0.70) CASP3CASP7CASP6CASP1CASP4
SCHEMBL18954440 0.83 ALDH1A1 (1.00) CASP3CASP7CASP6CASP1CASP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000038636-A1 AGENT FOR DYING KERATIN FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-07-06 WO claimed
CN-111423421-B Oxidized indole-substituted gamma-butenolide derivative and preparation method and application thereof 中山大学 2021-09-03 CN disclosed
CN-111423421-A Oxidized indole-substituted gamma-butenolide derivative and preparation method and application thereof 中山大学 2020-07-17 CN disclosed
WO-2000038636-A1 AGENT FOR DYING KERATIN FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-07-06 WO disclosed