SCHEMBL28026201

SCHEMBL28026201

O=C1C(=O)N(Cc2ccccc2Cl)c2ccc([N+](=O)[O-])cc21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.73
CASP3 P42574 2/20 0.73
CASP4 P49662 2/20 0.73
CASP7 P55210 2/20 0.73
CASP9 P55211 2/20 0.73
CASP6 P55212 2/20 0.73
CASP8 Q14790 1/20 0.73
CHRM5 P08912 2/20 0.58
ACHE P22303 2/20 0.58
ALDH1A1 P00352 3/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
CA12 O43570 5/20 0.55
CA1 P00915 5/20 0.55
CA2 P00918 5/20 0.55
CA9 Q16790 5/20 0.55
KDM1A O60341 1/20 0.50
ALDH2 P05091 2/20 0.49
ALDH3A1 P30838 2/20 0.49
MEN1 O00255 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28026202 0.85 ALDH1A1 (0.65) CASP1CASP3CASP4CASP7CASP9
SCHEMBL8019337 0.85 CASP3 (1.00) CASP1CASP3CASP4CASP7CASP9
SCHEMBL18954527 0.83 CASP1 (0.70) CASP1CASP3CASP4CASP7CASP9
SCHEMBL9904848 0.82 ALDH3A1 (0.72) CHRM5ALDH1A1CA12CA1CA2
SCHEMBL8019897 0.81 CASP3 (0.79) CASP1CASP3CASP4CASP7CASP9
SCHEMBL5659567 0.80 ALDH1A1 (0.71) CHRM5ACHEALDH1A1CA12CA1
SCHEMBL5659656 0.80 ACHE (0.66) CHRM5ACHEALDH1A1CA12CA1
SCHEMBL18954802 0.79 CHRM5 (0.60) CASP3CASP7CASP6CHRM5ACHE
SCHEMBL4609842 0.79 CES1 (0.66) CHRM5ACHEALDH1A1ALDH2ALDH3A1
SCHEMBL18954800 0.78 CHRM5 (0.58) CASP3CASP7CASP6CHRM5ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104829608-B A kind of cumarin thiazole indolone type compound and its preparation method and purposes 吉首大学 2017-06-30 CN disclosed
CN-104829608-A Coumarin-thiazole-indolone compounds, and preparation method and application thereof UNIV JISHOU 2015-08-12 CN disclosed