SCHEMBL8020187

SCHEMBL8020187

COC(=O)CN(C(=O)[C@@H](CCc1ccccc1)CSC(C)=O)c1ccc(OCc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
CACNA1C Q13936 1/20 0.44
MAOB P27338 5/20 0.43
KCNH2 Q12809 1/20 0.40
PTPN1 P18031 1/20 0.40
MAOA P21397 2/20 0.39
PLA2G4B P0C869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010485 0.93 ALDH1A1 (0.50) ALDH1A1CYP1A2MAOBPTPN1
SCHEMBL8020571 0.92 ALDH1A1 (0.51) ALDH1A1CYP1A2MAOBPTPN1
SCHEMBL8010570 0.90 ALDH1A1 (0.48) MEN1KMT2AALDH1A1CYP1A2MAOB
SCHEMBL8026762 0.89 ALDH1A1 (0.47) ALDH1A1CYP1A2MAOBPTPN1
SCHEMBL8020417 0.88 ALDH1A1 (0.46) ALDH1A1CYP1A2MAOBPTPN1
SCHEMBL8026201 0.88 ALDH1A1 (0.46) MEN1KMT2AALDH1A1MAPTMAOB
SCHEMBL8010401 0.87 ALDH1A1 (0.45) MEN1KMT2AALDH1A1MAPTMAOB
SCHEMBL8021208 0.87 ALDH1A1 (0.46) ALDH1A1CYP1A2MAOBKCNH2PTPN1
SCHEMBL8024218 0.86 ALDH1A1 (0.44) ALDH1A1CYP1A2MAOBPTPN1
SCHEMBL8026970 0.84 GPR132 (0.43) MEN1KMT2AALDH1A1MAPK1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed