SCHEMBL8026762

SCHEMBL8026762

COC(=O)CN(C(=O)C(CCc1ccccc1)CSC(C)=O)c1ccc(OCc2ccc(N(C)C)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
NOX1 Q9Y5S8 1/20 0.47
MAOB P27338 2/20 0.44
PTPN1 P18031 1/20 0.43
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
MLYCD O95822 1/20 0.40
MMP12 P39900 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABCC3 O15438 1/20 0.39
NR1I2 O75469 1/20 0.39
ABCB11 O95342 1/20 0.39
NR3C1 P04150 1/20 0.39
RARG P13631 1/20 0.39
CNR1 P21554 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010485 0.96 ALDH1A1 (0.50) ALDH1A1NOX1MAOBPTPN1LTB4R
SCHEMBL8020571 0.95 ALDH1A1 (0.51) ALDH1A1NOX1MAOBPTPN1MLYCD
SCHEMBL8010570 0.94 ALDH1A1 (0.48) ALDH1A1MAOBPTPN1MLYCDMMP12
SCHEMBL8026871 0.93 PPARG (0.43) ALDH1A1NOX1MAOBPTPN1MLYCD
SCHEMBL8020417 0.92 ALDH1A1 (0.46) ALDH1A1MAOBPTPN1LTB4RLTB4R2
SCHEMBL8026201 0.91 ALDH1A1 (0.46) ALDH1A1MAOBPTPN1ALOX5
SCHEMBL8010401 0.91 ALDH1A1 (0.45) ALDH1A1NOX1MAOBPTPN1
SCHEMBL8021208 0.90 ALDH1A1 (0.46) ALDH1A1NOX1MAOBPTPN1MLYCD
SCHEMBL8024218 0.90 ALDH1A1 (0.44) ALDH1A1MAOBPTPN1MLYCDMMP12
SCHEMBL8020187 0.89 MEN1 (0.44) ALDH1A1MAOBPTPN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed