SCHEMBL8020707

SCHEMBL8020707

Cc1cc(-c2ccc(Oc3ccc(N)cc3)c(C)c2)ccc1Oc1ccc(N)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
TEAD4 Q15561 1/20 0.50
MAPT P10636 5/20 0.48
TDP1 Q9NUW8 3/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 2/20 0.48
TSHR P16473 2/20 0.48
HPGD P15428 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NCOA1 Q15788 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MITF O75030 1/20 0.44
GAA P10253 1/20 0.44
GFER P55789 1/20 0.44
NLRP1 Q9C000 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915293 0.96 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL2989217 0.89 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL1155719 0.88 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL31457276 0.88 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL1810759 0.86 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL29510593 0.86 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL2992329 0.86 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL11528953 0.85 TEAD4 (0.61) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL31457328 0.84 NCOA1 (0.50) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL3003478 0.84 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069278-A Aromatic diamines and polyimides based on 4,4'-bis-(4-aminophenoxy)-2,2' or 2,2',6,6'-substituted biphenyl THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 2000-05-30 US disclosed
US-6037499-A 4,4'-BIS(4-AMINOPHENOXY),2,2',6,6'-SUBSTITUTED BIPHENYL RADICALS EXHIBITING NONCOPLANAR CONFORMATION FOR ENHANCED SOLUBILITY; POLYIMIDES MADE THEREFROM HAVE GOOD PROCESSABILITY AND HIGH GLASS TRANSITION TEMPERATURE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 2000-03-14 US disclosed
US-5939521-A THERMOPLASTIC POLYIMIDES DERIVED FROM THE AROMATIC DIAMINES OF THIS INVENTION ARE CHARACTERIZED AS HAVING A HIGH GLASS TRANSITION TEMPERATURE, GOOD MECHANICAL PROPERTIES AND IMPROVED PROCESSABILITY IN THE MANUFACTURE OF ADHESIVES, THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1999-08-17 US disclosed
US-5844065-A 2,2'-dimethyl-4,4'-bis (4-aminophenoxy) biphenyl, and polymers prepared therefrom by polycondensation NATIONAL SCIENCE COUNCIL (TW) 1998-12-01 US disclosed
US-5650463-A Carbon fiber-reinforced polimide resin composition MITSUI TOATSU CHEMICALS, INC. (JP) 1997-07-22 US disclosed
US-5554765-A HEAT RESISTANCE MITSUI TOATSU CHEMICALS, INC. (JP) 1996-09-10 US disclosed
EP-0523240-B1 BISIMIDE COMPOUNDS, POLYIMIDE RESIN COMPOSITION PREPARED THEREFROM, AND CARBON FIBER-REINFORCED POLYIMIDE RESIN COMPOSITION MITSUI TOATSU CHEMICALS (JP) 1996-03-20 EP disclosed
US-5457154-A Melt processability MITSUI TOATSU CHEMICALS, INC. (JP) 1995-10-10 US disclosed
EP-0523240-A1 BISIMIDE COMPOUNDS, POLYIMIDE RESIN COMPOSITION PREPARED THEREFROM, AND CARBON FIBER-REINFORCED POLYIMIDE RESIN COMPOSITION MITSUI TOATSU CHEMICALS, Inc. (JP) 1993-01-20 EP disclosed