SCHEMBL8021371

SCHEMBL8021371

COC(=O)CNc1cccc(Cc2ccc(OC)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SAE1 Q9UBE0 1/20 0.51
UBA2 Q9UBT2 1/20 0.51
MTNR1A P48039 2/20 0.49
MTNR1B P49286 2/20 0.49
LTA4H P09960 1/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
PPARA Q07869 1/20 0.46
NLRP3 Q96P20 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
HTT P42858 1/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026490 0.89 AKR1C3 (0.44) MTNR1AMTNR1BLTA4HSMN1; SMN2GAA
SCHEMBL8026213 0.88 GAA (0.43) SAE1UBA2MTNR1AMTNR1BLTA4H
SCHEMBL9780049 0.81 MTNR1A (0.61) MTNR1AMTNR1BNLRP3SMN1; SMN2MAPT
SCHEMBL8020284 0.81 GRK2 (0.57) MTNR1AMTNR1BCA12CA1CA2
Hydrochloric Acid SCHEMBL5109957 0.80 MTNR1A (0.60) MTNR1AMTNR1BNLRP3SMN1; SMN2MAPT
SCHEMBL9795665 0.79 MTNR1A (0.41) MTNR1AMTNR1BCA12CA1CA2
Hydrochloric Acid SCHEMBL28230977 0.78 LTA4H (0.59) SAE1UBA2MTNR1AMTNR1BLTA4H
SCHEMBL9779998 0.77 MAPT (0.59) SAE1UBA2CA12CA1CA2
SCHEMBL9779958 0.77 SIRT2 (0.45) NLRP3GAA
Hydrochloric Acid SCHEMBL5122021 0.76 MAPT (0.57) SAE1UBA2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed