SCHEMBL8026490

SCHEMBL8026490

COC(=O)CNc1cccc(Cc2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.44
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
LTA4H P09960 1/20 0.43
USP2 O75604 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.42
HIF1A Q16665 2/20 0.42
FFAR1 O14842 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026213 0.90 GAA (0.43) MTNR1AMTNR1BRAB9ASMN1; SMN2KDM4E
SCHEMBL8021371 0.89 SAE1 (0.51) MTNR1AMTNR1BRAB9ASMN1; SMN2NPC1
SCHEMBL9795665 0.83 MTNR1A (0.41) AKR1C3MTNR1AMTNR1BUSP2SIRT2
SCHEMBL9779958 0.82 SIRT2 (0.45) GAASIRT2FFAR1
SCHEMBL658053 0.82 LMNA (0.54) RAB9ASMN1; SMN2KDM4ENPC1ALDH1A1
SCHEMBL8009616 0.80 FFAR1 (0.58) LTA4HSIRT2FFAR1
Benzene SCHEMBL28330086 0.80 LMNA (0.53) AKR1C3RAB9ASMN1; SMN2KDM4ENPC1
Hydrochloric Acid SCHEMBL76327 0.80 LMNA (0.53) AKR1C3RAB9ASMN1; SMN2KDM4ENPC1
SCHEMBL8021547 0.79 ALDH1A1 (0.55) RAB9ASMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL2092346 0.78 SMN1; SMN2 (0.54) RAB9ASMN1; SMN2NPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed
EP-0934262-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-08-11 EP disclosed
WO-1998017639-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1998-04-30 WO disclosed