SCHEMBL8022360

SCHEMBL8022360

NC(=O)C#Cc1cccs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.44
GRM5 P41594 2/20 0.42
ALDH1A1 P00352 3/20 0.39
POLB P06746 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
ERN1 O75460 1/20 0.38
DAO P14920 1/20 0.38
GSK3B P49841 1/20 0.37
HDAC1 Q13547 1/20 0.35
ALOX5 P09917 1/20 0.35
HPGD P15428 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
F2 P00734 1/20 0.34
PRSS1 P07477 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18104962 0.83 FFAR1 (0.46) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL3946468 0.82 FFAR1 (0.49) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL1159454 0.80 GRM5 (0.46) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL28454253 0.77 RAB9A (0.50) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL7202747 0.76 HSP90AA1 (0.49) FFAR1GRM5ALDH1A1NPC1RAB9A
SCHEMBL28502889 0.76 FFAR1 (0.44) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL20089251 0.76 GRM5 (0.42) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL9329997 0.75 GRM5 (0.40) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL2491796 0.75 GRM5 (0.55) FFAR1GRM5ALDH1A1POLBNPC1
SCHEMBL7199097 0.73 SMN1; SMN2 (0.37) FFAR1GRM5ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023274246-A1 AMIDE COMPOUND AND USE THEREOF 成都分迪药业有限公司 2023-01-05 WO disclosed
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
US-5917038-A REACTING PROPIOLAMIDE WITH ACTIVATED AROMATIC RING IN THE PRESENCE OF A PALLADIUM CATALYST ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed