SCHEMBL8022584

SCHEMBL8022584

BrCc1cccc(C2OCCO2)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TRPA1 O75762 1/20 0.37
TSHR P16473 1/20 0.37
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.31
HTR2A P28223 2/20 0.30
HTR2C P28335 2/20 0.30
HTR2B P41595 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL334828 0.82 MEN1 (0.40) ALDH1A1HTTSMN1; SMN2TRPA1TSHR
SCHEMBL232609 0.82 SLC5A2 (0.35) ALDH1A1HTTSMN1; SMN2TSHRMEN1
SCHEMBL5604860 0.81 NCF1 (0.44) ALDH1A1HTTSMN1; SMN2
SCHEMBL6517254 0.81 CHRNB4 (0.45) ALDH1A1HTTSMN1; SMN2TSHR
SCHEMBL6517744 0.81 FOLH1 (0.38) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL11941052 0.81 SMN1; SMN2 (0.49) ALDH1A1HTTSMN1; SMN2LMNARAB9A
SCHEMBL9520126 0.80 SIGMAR1 (0.35) ALDH1A1HTTSMN1; SMN2TSHRMEN1
SCHEMBL189832 0.79 TRPA1 (0.38) ALDH1A1TRPA1TSHR
SCHEMBL6513629 0.79 ALDH1A1 (0.36) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL9262464 0.79 ALDH1A1 (0.39) ALDH1A1HTTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143170-B For treating the aromatic compounds of pulmonary fibrosis, liver fibrosis, fibrosis of skin and cardiac fibrosis being substituted 普罗米蒂克医药SMT有限公司 2019-11-08 CN disclosed
WO-2000049020-A2 NOVEL EPOTHILON DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR PHARMACEUTICAL APPLICATION SCHERING AKTIENGESELLSCHAFT (DE) 2000-08-24 WO disclosed
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed