SCHEMBL8023112

SCHEMBL8023112

CC(C)(Br)C(=O)Nc1ccccc1NC(=O)C(C)(C)Br

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.53
PDK1 Q15118 10/20 0.51
PDK2 Q15119 10/20 0.51
PDK3 Q15120 10/20 0.51
PDK4 Q16654 10/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
RECQL P46063 1/20 0.50
HTT P42858 1/20 0.47
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1555152 0.88 GAA (0.54) CETPPDK1PDK2PDK3PDK4
SCHEMBL19280535 0.88 PDK1 (0.68) CETPPDK1PDK2PDK3PDK4
SCHEMBL18458382 0.86 PDK1 (0.68) PDK1PDK2PDK3PDK4SMN1; SMN2
SCHEMBL5706504 0.84 CETP (0.71) CETPPDK1PDK2PDK3PDK4
SCHEMBL7421740 0.82 PDK1 (0.68) PDK1PDK2PDK3PDK4SMN1; SMN2
SCHEMBL436619 0.80 PDK1 (0.61) PDK1PDK2PDK3PDK4SMN1; SMN2
SCHEMBL8032793 0.80 CETP (0.52) CETPPDK1PDK2PDK3PDK4
SCHEMBL30797039 0.79 PDK1 (0.50) CETPPDK1PDK2PDK3PDK4
SCHEMBL4675699 0.79 PDK1 (0.50) CETPPDK1PDK2PDK3PDK4
SCHEMBL24251779 0.78 BLM (0.42) CETPPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127536-A Synthesis of a tetraamido macrocycle ligand THE CLOROX COMPANY (US) 2000-10-03 US disclosed