SCHEMBL24251779

SCHEMBL24251779

CC(C)(Br)C(=O)Nc1ccc[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 3/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NAPRT Q6XQN6 1/20 0.41
CDC25A P30304 1/20 0.40
CDC25B P30305 1/20 0.40
ALPL P05186 1/20 0.40
DAO P14920 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CETP P11597 1/20 0.39
PRSS1 P07477 1/20 0.39
TMPRSS15 P98073 1/20 0.39
PDK1 Q15118 3/20 0.39
PDK2 Q15119 3/20 0.39
PDK3 Q15120 3/20 0.39
PDK4 Q16654 3/20 0.39
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493519 0.81 JAK2 (0.51) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL6826283 0.79 ALDH1A1 (0.50) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL8023112 0.78 CETP (0.53) TSHRALDH1A1CETPPDK1PDK2
SCHEMBL6286018 0.78 RAB9A (0.52) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL16794593 0.77 NAPRT (0.52) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL3431388 0.75 GAA (0.47) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL26790018 0.75 ALDH1A1 (0.52) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL20033714 0.73 BLM (0.44) BLMTSHRALDH1A1HSD17B10NAPRT
SCHEMBL29623640 0.72 KCNMA1 (0.55) ALDH1A1HSD17B10CDC25ACDC25BGSK3A
SCHEMBL19280535 0.72 PDK1 (0.68) ALDH1A1CETPPDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed