SCHEMBL8023307

SCHEMBL8023307

CC1(C)C(=O)N(c2ccccc2)C(=O)N1Cc1ccccc1Oc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAS2R8 Q9NYW2 10/20 0.47
FAAH O00519 1/20 0.43
IGF1R P08069 1/20 0.41
RIPK1 Q13546 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
CYP19A1 P11511 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ELANE P08246 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
HRH1 P35367 1/20 0.38
TNF P01375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021401 0.95 TAS2R8 (0.46) TAS2R8FAAHIGF1RRIPK1SLC6A2
SCHEMBL8010593 0.93 TAS2R8 (0.44) TAS2R8FAAHIGF1RSLC6A4
SCHEMBL8019464 0.93 TAS2R8 (0.44) TAS2R8FAAHIGF1RRIPK1SLC6A2
SCHEMBL8023309 0.93 TAS2R8 (0.46) TAS2R8FAAHIGF1RSLC6A4CYP19A1
SCHEMBL8020845 0.93 TAS2R8 (0.44) TAS2R8FAAHRIPK1SLC6A2SLC6A4
SCHEMBL12873224 0.92 TAS2R8 (0.48) TAS2R8FAAHIGF1RSLC6A2SLC6A4
SCHEMBL8006275 0.92 TAS2R8 (0.44) TAS2R8FAAHIGF1RRIPK1SLC6A2
SCHEMBL8027028 0.92 HTR2A (0.47) TAS2R8FAAHIGF1RSLC6A2SLC6A4
SCHEMBL8024739 0.91 TAS2R8 (0.43) TAS2R8FAAHIGF1RHDAC1HDAC6
SCHEMBL8010523 0.91 TAS2R8 (0.43) TAS2R8FAAHIGF1RCYP19A1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed
WO-2009097998-A1 ARYLCHALCOGENO-ARYLALKYL-SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046185-A1 Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof PGC, LIPC, CEL TAS2R8 318/4885FAAH 1395/4885IGF1R 645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.