SCHEMBL8041285

SCHEMBL8041285

COc1cc(Cl)c(C(=O)NC(=O)NC(C)(C)C)cc1OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 4/20 0.51
HPGD P15428 3/20 0.51
SMPD1 P17405 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CTSV O60911 2/20 0.47
CTSL P07711 2/20 0.47
EGFR P00533 1/20 0.47
LMNA P02545 2/20 0.45
SRD5A1 P18405 1/20 0.45
SRD5A2 P31213 1/20 0.45
PYGL P06737 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 2/20 0.44
GAA P10253 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025544 0.85 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDSMPD1HDAC1
SCHEMBL8039095 0.85 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDSMPD1HDAC1
SCHEMBL8037235 0.85 SMPD1 (0.45) ALDH1A1KDM4EHPGDSMPD1HDAC1
SCHEMBL8037213 0.83 MEN1 (0.51) ALDH1A1SMPD1HDAC1HDAC8HDAC6
SCHEMBL8039242 0.83 SMPD1 (0.54) ALDH1A1KDM4EHPGDSMPD1HDAC1
SCHEMBL8039089 0.82 MTNR1A (0.49) HPGDSMPD1HDAC1HDAC8HDAC6
SCHEMBL8025539 0.82 MTNR1A (0.48) HPGDSMPD1HDAC1HDAC8HDAC6
SCHEMBL8037325 0.82 NPC1 (0.47) ALDH1A1SMPD1HDAC1HDAC8HDAC6
SCHEMBL8037216 0.81 SGMS2 (0.58) ALDH1A1SMPD1HDAC1HDAC8HDAC6
SCHEMBL8035583 0.81 SGMS2 (0.58) ALDH1A1SMPD1HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed