SCHEMBL8026871

SCHEMBL8026871

COC(=O)CN(C(=O)[C@@H](CCc1ccccc1)CSC(C)=O)c1ccc(OCCc2ccc(N(C)C)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.43
MLYCD O95822 1/20 0.40
FFAR1 O14842 1/20 0.39
ALDH1A1 P00352 1/20 0.39
NOX1 Q9Y5S8 1/20 0.38
LTA4H P09960 2/20 0.38
MAOB P27338 1/20 0.36
PTPN1 P18031 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026762 0.93 ALDH1A1 (0.47) MLYCDFFAR1ALDH1A1NOX1MAOB
SCHEMBL8010485 0.89 ALDH1A1 (0.50) MLYCDFFAR1ALDH1A1NOX1MAOB
SCHEMBL8020571 0.88 ALDH1A1 (0.51) MLYCDALDH1A1NOX1MAOBPTPN1
SCHEMBL8010570 0.87 ALDH1A1 (0.48) MLYCDFFAR1ALDH1A1MAOBPTPN1
SCHEMBL8020417 0.85 ALDH1A1 (0.46) MLYCDFFAR1ALDH1A1MAOBPTPN1
SCHEMBL8026201 0.84 ALDH1A1 (0.46) ALDH1A1MAOBPTPN1
SCHEMBL8024569 0.84 MLYCD (0.45) MLYCDALDH1A1
SCHEMBL8010401 0.84 ALDH1A1 (0.45) ALDH1A1NOX1LTA4HMAOBPTPN1
SCHEMBL8021208 0.83 ALDH1A1 (0.46) MLYCDALDH1A1NOX1MAOBPTPN1
SCHEMBL8024218 0.83 ALDH1A1 (0.44) MLYCDFFAR1ALDH1A1MAOBPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed