SCHEMBL8028834

SCHEMBL8028834

CCC(=O)C(=Cc1cccc(C#N)c1)C(=O)CC

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.59
CD274 Q9NZQ7 1/20 0.59
FBP1 P09467 3/20 0.55
P4HB P07237 13/20 0.48
GRIN2D O15399 2/20 0.43
GRIN3B O60391 2/20 0.43
GRIN1 Q05586 2/20 0.43
GRIN2A Q12879 2/20 0.43
GRIN2B Q13224 2/20 0.43
GRIN2C Q14957 2/20 0.43
GRIN3A Q8TCU5 2/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Balazipone SCHEMBL636109 0.84 PDCD1 (0.55) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL8039347 0.80 FBP1 (0.54) FBP1P4HBGSK3B
SCHEMBL9475839 0.80 PDCD1 (0.51) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL9475845 0.80 PDCD1 (0.51) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL10375509 0.79 PDCD1 (0.71) PDCD1CD274FBP1
SCHEMBL10848993 0.79 PDCD1 (0.71) PDCD1CD274FBP1
SCHEMBL3115027 0.78 AKR1C3 (0.59) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL6981746 0.78 AKR1C3 (0.59) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL28372992 0.78 AKR1C3 (0.59) PDCD1CD274FBP1P4HBGRIN2D
SCHEMBL6947906 0.77 PDCD1 (0.54) PDCD1CD274FBP1P4HBGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP claimed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US claimed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP claimed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-5292771-A Treating inflammatory bowel disease ORION-YHTYMA OY (FI) 1994-03-08 US disclosed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP disclosed