SCHEMBL9475845

SCHEMBL9475845

CC(=O)C(=Cc1cccc(C#N)c1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.51
CD274 Q9NZQ7 1/20 0.51
FBP1 P09467 3/20 0.50
GLO1 Q04760 1/20 0.46
P4HB P07237 8/20 0.45
KDM4E B2RXH2 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
HTT P42858 1/20 0.43
GRIN2D O15399 2/20 0.42
GRIN3B O60391 2/20 0.42
GRIN1 Q05586 2/20 0.42
GRIN2A Q12879 2/20 0.42
GRIN2B Q13224 2/20 0.42
GRIN2C Q14957 2/20 0.42
GRIN3A Q8TCU5 2/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9475839 1.00 PDCD1 (0.51) PDCD1CD274FBP1GLO1P4HB
Balazipone SCHEMBL636109 0.92 PDCD1 (0.55) PDCD1CD274FBP1GLO1P4HB
SCHEMBL6981746 0.86 AKR1C3 (0.59) PDCD1CD274FBP1P4HBKDM4E
SCHEMBL28372992 0.86 AKR1C3 (0.59) PDCD1CD274FBP1P4HBKDM4E
SCHEMBL3115027 0.86 AKR1C3 (0.59) PDCD1CD274FBP1P4HBKDM4E
SCHEMBL9842162 0.85 GLO1 (0.46) PDCD1CD274GLO1KDM4EHTT
SCHEMBL9842160 0.85 GLO1 (0.46) PDCD1CD274GLO1KDM4EHTT
SCHEMBL6947906 0.84 PDCD1 (0.54) PDCD1CD274FBP1GLO1P4HB
SCHEMBL6947909 0.84 PDCD1 (0.54) PDCD1CD274FBP1GLO1P4HB
SCHEMBL10848993 0.81 PDCD1 (0.71) PDCD1CD274FBP1GLO1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202330-A Hypotensive and cardiovascular agent, reduces blood pressure in mammals E. R. SQUIBB & SONS, INC. (US) 1993-04-13 US disclosed
EP-0204317-A2 2-Thio or oxo-4-aryl or heterocyclo-1,5(2H)-pyrimidinedicarboxylic acid diesters and 3-acyl-5-pyrimidinecarboxylic acids and esters E.R. Squibb & Sons, Inc. (US) 1986-12-10 EP disclosed