SCHEMBL8029433

SCHEMBL8029433

Cc1cc2cc(C#N)ccc2n1CC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPK1 P28482 1/20 0.45
STAT3 P40763 1/20 0.45
CCR2 P41597 1/20 0.44
BRPF1 P55201 1/20 0.43
CNR1 P21554 6/20 0.41
CCR9 P51686 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KMO O15229 1/20 0.40
SMARCA2 P51531 1/20 0.40
LMNA P02545 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3005494 0.80 PTGDR2 (0.47) ALDH1A1L3MBTL1KDM4EGAAKMO
SCHEMBL10054048 0.80 BRPF1 (0.50) ALDH1A1BRPF1CNR1KDM4EGAA
SCHEMBL3785498 0.80 SCN7A (0.56) NTRK1ALDH1A1MAPK1STAT3CCR2
SCHEMBL2591249 0.78 KDM4E (0.49) ALDH1A1CCR2KDM4E
SCHEMBL1467597 0.78 CCR2 (0.54) CCR2KMO
SCHEMBL1251025 0.78 CCR2 (0.47) ALDH1A1CCR2BRPF1L3MBTL1KDM4E
SCHEMBL7958147 0.77 NTRK1 (0.57) NTRK1CCR2BRPF1CNR1CCR9
SCHEMBL16709583 0.76 PTGDR2 (0.50) ALDH1A1MAPK1STAT3L3MBTL1KDM4E
SCHEMBL3067363 0.75 L3MBTL1 (0.64) ALDH1A1CCR2L3MBTL1KDM4EMAPT
SCHEMBL27990361 0.74 CCR2 (0.50) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043257-A ANTICOAGULANT; PYRIDINE SUBSTITUTED INDAZOLE COMPOUND E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-03-28 US disclosed
US-5886191-A ANTICOAGULANTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-23 US disclosed