SCHEMBL16709583

SCHEMBL16709583

Cc1ccc2c(c1)c1cc(C#N)ccc1n2CC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 16/20 0.50
AKR1B1 P15121 7/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPK1 P28482 1/20 0.50
STAT3 P40763 1/20 0.50
CYP2C9 P11712 2/20 0.47
KDM4E B2RXH2 2/20 0.45
POLB P06746 1/20 0.45
HSD17B10 Q99714 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15486120 0.83 TSPO (0.45) PTGDR2AKR1B1ALDH1A1MAPK1STAT3
SCHEMBL1406080 0.80 PTGDR2 (0.75) PTGDR2AKR1B1ALDH1A1MAPK1STAT3
SCHEMBL1386238 0.79 PTGDR2 (0.74) PTGDR2AKR1B1ALDH1A1MAPK1STAT3
SCHEMBL15486750 0.78 PTGDR2 (0.53) PTGDR2AKR1B1CYP2C9KDM4EPOLB
SCHEMBL15599705 0.78 PTGDR2 (0.53) PTGDR2AKR1B1CYP2C9KDM4EPOLB
SCHEMBL15733080 0.77 MARK4 (0.57) PTGDR2AKR1B1CYP2C9KDM4EPOLB
SCHEMBL20046019 0.76 RORA (0.56) ALDH1A1
SCHEMBL8029433 0.76 NTRK1 (0.46) ALDH1A1MAPK1STAT3KDM4EL3MBTL1
SCHEMBL18055752 0.76 ALDH1A1 (0.47) ALDH1A1MAPK1KDM4E
SCHEMBL19368919 0.75 PTGDR2 (0.63) PTGDR2AKR1B1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015070237-A1 NEUROPROTECTIVE CHEMICALS AND METHODS FOR IDENTIFYING AND USING SAME BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-05-14 WO disclosed