SCHEMBL8032196

SCHEMBL8032196

CC[C@@H](NC(=O)c1ccc(NCc2ncc(F)cc2F)c(N)c1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
HDAC3 O15379 4/20 0.43
HDAC1 Q13547 4/20 0.43
HDAC2 Q92769 4/20 0.43
NCOR2 Q9Y618 4/20 0.43
PTGER4 P35408 1/20 0.43
SLC6A9 P48067 1/20 0.42
TACR3 P29371 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033972 0.86 PPARG (0.57) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8038556 0.84 PPARG (0.61) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8032177 0.84 PPARG (0.60) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8034344 0.83 PPARG (0.54) PPARGHDAC3HDAC1HDAC2NCOR2
SCHEMBL4538730 0.83 PPARG (0.57) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4537762 0.81 PPARG (0.48) PPARGHDAC1
SCHEMBL4540765 0.81 MEN1 (0.52) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4538247 0.81 PPARG (0.59) PPARG
SCHEMBL4537201 0.80 PPARG (0.57) PPARGCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8032490 0.79 PPARG (0.55) PPARGHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed