SCHEMBL8032341

SCHEMBL8032341

Cc1cc(-n2nnnc2Sc2ncc([N+](=O)[O-])s2)sc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
TLR9 Q9NR96 3/20 0.46
KMT2A Q03164 3/20 0.46
AGTR1 P30556 2/20 0.46
MEN1 O00255 2/20 0.46
MAPK8 P45983 9/20 0.44
MAPK9 P45984 9/20 0.44
MAPK10 P53779 2/20 0.44
ALDH1A1 P00352 5/20 0.40
MAPT P10636 3/20 0.40
HTT P42858 3/20 0.40
MAPK1 P28482 3/20 0.40
S1PR4 O95977 2/20 0.40
S1PR1 P21453 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HSP90AA1 P07900 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050814 0.83 MAPK8 (0.44) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8043929 0.82 MAPK8 (0.47) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8034482 0.81 ALDH1A1 (0.36) KMT2AALDH1A1MAPTHTTMAPK1
SCHEMBL8043586 0.79 NPC1 (0.46) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8050613 0.79 MAPT (0.46) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8047788 0.79 LMNA (0.31) KMT2AALDH1A1MAPTHTTMAPK1
SCHEMBL8046585 0.79 RXRA (0.43) KMT2AMEN1ALDH1A1MAPTHTT
SCHEMBL8042307 0.78 MAPK8 (0.52) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8046704 0.77 ALDH1A1 (0.60) NPC1RAB9ATLR9KMT2AAGTR1
SCHEMBL8048172 0.77 MITF (0.47) NPC1RAB9ATLR9KMT2AAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed