SCHEMBL8032445

SCHEMBL8032445

O=C(O)Cn1nnnc1Sc1nc2ccccc2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
HPGD P15428 5/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
TSHR P16473 3/20 0.50
POLB P06746 3/20 0.50
MAPK1 P28482 3/20 0.50
HSD17B10 Q99714 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
APEX1 P27695 1/20 0.47
RECQL P46063 1/20 0.47
AKR1B1 P15121 1/20 0.47
MAPT P10636 3/20 0.45
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050220 0.84 MAPT (0.43) ALDH1A1HPGDSMN1; SMN2POLBHSD17B10
SCHEMBL8045150 0.83 ALDH1A1 (0.52) ALDH1A1HPGDSMN1; SMN2TSHRPOLB
SCHEMBL8044261 0.83 ALDH1A1 (0.50) ALDH1A1HPGDSMN1; SMN2TSHRPOLB
SCHEMBL8034157 0.82 AKR1B1 (0.42) ALDH1A1HPGDSMN1; SMN2MAPK1AKR1B1
SCHEMBL8050578 0.81 ALDH1A1 (0.49) ALDH1A1HPGDSMN1; SMN2TSHRPOLB
SCHEMBL8044630 0.81 PDK1 (0.53) ALDH1A1HPGDSMN1; SMN2TSHRMAPK1
SCHEMBL8043976 0.81 KDM4E (0.43) ALDH1A1HPGDSMN1; SMN2TSHRHSD17B10
SCHEMBL8049808 0.81 SMN1; SMN2 (0.50) ALDH1A1HPGDSMN1; SMN2TSHRPOLB
SCHEMBL8032720 0.79 HSP90AA1 (0.53) ALDH1A1HPGDSMN1; SMN2TSHRPOLB
SCHEMBL8048335 0.79 RAB9A (0.45) ALDH1A1HPGDSMN1; SMN2TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed