SCHEMBL8032578

SCHEMBL8032578

CN(C)c1ccc(-c2nc(-c3ccc(O)cc3)[nH]c2-c2ccc(N(C)C)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 2/20 0.76
ALOX5 P09917 2/20 0.65
MAPT P10636 5/20 0.59
TP53 P04637 4/20 0.59
MAPK14 Q16539 4/20 0.59
MAPK13 O15264 3/20 0.59
MAPK12 P53778 3/20 0.59
MAPK11 Q15759 3/20 0.59
RAF1 P04049 2/20 0.59
BRAF P15056 2/20 0.59
GCGR P47871 2/20 0.59
CSNK1D P48730 2/20 0.58
CSNK1E P49674 2/20 0.58
KDM4E B2RXH2 1/20 0.58
CIT O14578 1/20 0.58
GAK O14976 1/20 0.58
RIPK2 O43353 1/20 0.58
BRD4 O60885 1/20 0.58
GMNN O75496 1/20 0.58
PRKD3 O94806 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010209 0.87 NOX1 (0.76) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL1071183 0.86 NOX1 (1.00) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL5622957 0.85 ALOX5 (0.87) NOX1ALOX5MAPTMAPK14MAPK13
SCHEMBL6468252 0.85 NOX1 (0.76) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL8797410 0.83 NOX1 (0.72) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL12103631 0.83 NOX1 (0.64) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL6467424 0.82 NOX1 (0.72) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL12103613 0.82 NOX1 (0.63) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL14336058 0.82 NOX1 (0.78) NOX1ALOX5MAPTTP53MAPK14
SCHEMBL9619859 0.81 MAPK13 (0.85) NOX1ALOX5MAPTTP53MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347139-A2 Imidazole leuco dye composition containing 4'-hydroxyacetanilide diagnostic kit and method using same EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1989-12-20 EP claimed
US-4089747-A OXIDATION OF DYE-PROVIDING MATERIALS, A SULFONYL HYDRAZONE AND A COUPLER OR A TRIARYLIMIDAZOLE EASTMAN KODAK COMPANY (US) 1978-05-16 US claimed
EP-0603954-B1 Immunoassay using a 4-hydroxy or 4-alkoxyarylacetamide as stabilizer JOHNSON & JOHNSON CLIN DIAG (US) 2000-03-08 EP disclosed
EP-0603953-B1 Use of 4' of 5'-hydroxy and 4'- or 5'-alkoxy-substituted electron transfer agents in compositions, elements, test kits and analytical methods JOHNSON & JOHNSON CLIN DIAG (US) 1999-02-17 EP disclosed
US-5700826-A SENSITIZATION OF CANCER CELLS TO DRUG ONTOGEN CORPORATION (US) 1997-12-23 US disclosed
EP-0812829-A1 Substituted imidazoles as modulators of multi-drug resistance ONTOGEN CORPORATION (US) 1997-12-17 EP disclosed
EP-0431682-B1 Buffered wash composition, insolubilizing composition, test kits and method of use EASTMAN KODAK CO (US) 1995-02-01 EP disclosed
US-5372931-A Use of 4'-hydroxy- and 4'-alkoxy-substituted electron transfer agents in compositions, elements, test kits and analytical methods EASTMAN KODAK COMPANY (US) 1994-12-13 US disclosed
US-5372932-A Peroxidase-labeled immunoreactant; stabiliztion with a 4-hydroxy or 4-alkoxyarylacetamide EASTMAN KODAK COMPANY (US) 1994-12-13 US disclosed
EP-0308236-B1 Dye-providing composition, diagnostic test kit and their use in method for ligand determination using peroxidase labeled-receptor EASTMAN KODAK CO (US) 1994-11-23 EP disclosed
US-5366864-A Buffered wash composition, insolubilizing composition, test kits and method of use EASTMAN KODAK COMPANY (US) 1994-11-22 US disclosed
EP-0603953-A1 Use of 4' of 5'-hydroxy and 4'- or 5'-alkoxy-substituted electron transfer agents in compositions, elements, test kits and analytical methods Johnson & Johnson Clinical Diagnostics, Inc. (US) 1994-06-29 EP disclosed
EP-0603954-A2 Analytical element and immunoassay using a 4-hydroxy or 4-alkoxyarylacetamide as stabilizer Johnson & Johnson Clinical Diagnostics, Inc. (US) 1994-06-29 EP disclosed
US-5176999-A BUFFERED WASH COMPOSITION, INSOLUBILIZING COMPOSITION, TEST KITS AND METHOD OF USE EASTMAN KODAK COMPANY (US) 1993-01-05 US disclosed
US-5047318-A Detection Of Grampositive Bacteria EASTMAN KODAK COMPANY (US) 1991-09-10 US disclosed
US-5024935-A Determination of human chorionic gonadotropin EASTMAN KODAK COMPANY (US) 1991-06-18 US disclosed
EP-0431682-A2 Buffered wash composition, insolubilizing composition, test kits and method of use Johnson & Johnson Clinical Diagnostics, Inc. (US) 1991-06-12 EP disclosed
EP-0347139-A2 Imidazole leuco dye composition containing 4'-hydroxyacetanilide diagnostic kit and method using same EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1989-12-20 EP disclosed
EP-0308236-A2 Dye-providing composition, diagnostic test kit and their use in method for ligand determination using peroxidase labeled-receptor Johnson & Johnson Clinical Diagnostics, Inc. (US) 1989-03-22 EP disclosed
US-4089747-A OXIDATION OF DYE-PROVIDING MATERIALS, A SULFONYL HYDRAZONE AND A COUPLER OR A TRIARYLIMIDAZOLE EASTMAN KODAK COMPANY (US) 1978-05-16 US disclosed