SCHEMBL8034975

SCHEMBL8034975

O=C(O)c1nsc2nc3ccccc3n12.[Na]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 3/20 0.42
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
HIF1A Q16665 1/20 0.41
SMN1; SMN2 Q16637 6/20 0.41
TP53 P04637 2/20 0.41
MAOA P21397 1/20 0.41
CA12 O43570 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
RECQL P46063 2/20 0.40
CA1 P00915 1/20 0.40
ALDH1A1 P00352 4/20 0.40
MAPT P10636 3/20 0.39
HPGD P15428 2/20 0.39
MAPK1 P28482 2/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7483925 0.98 KDM4E (0.43) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7469069 0.85 MAOA (0.51) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7486338 0.84 KDM4E (0.47) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7474964 0.83 HSD17B10 (0.44) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7486359 0.81 NPC1 (0.45) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7484099 0.81 ADORA3 (0.43) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7485473 0.81 ALDH1A1 (0.49) KDM4EHSD17B10NPC1RAB9ASMN1; SMN2
SCHEMBL7484824 0.79 HPGD (0.44) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7485791 0.79 MAOA (0.40) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7485787 0.79 MAOA (0.40) KDM4EHSD17B10MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed
EP-0883606-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031893-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1997-09-04 WO disclosed