SCHEMBL8035110

SCHEMBL8035110

COc1cc(C(F)(F)F)c(C(=O)NC(=O)N(C(C)C)C2CCCCC2)cc1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 3/20 0.45
SGMS2 Q8NHU3 1/20 0.41
NPC1 O15118 2/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SMPD1 P17405 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
LMNA P02545 1/20 0.39
APP P05067 2/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
CYP19A1 P11511 1/20 0.37
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
PDE4A P27815 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025472 0.89 SGMS2 (0.42) TRPM8SGMS2NPC1PKMRAB9A
SCHEMBL8041224 0.88 SMPD1 (0.44) TRPM8NPC1PKMRAB9AALDH1A1
SCHEMBL8035618 0.84 APP (0.44) TRPM8NPC1PKMRAB9AMEN1
SCHEMBL8025476 0.83 SMPD1 (0.47) NPC1RAB9AMEN1KMT2ASMPD1
SCHEMBL8041228 0.82 SGMS2 (0.53) SGMS2NPC1RAB9AALDH1A1MEN1
SCHEMBL8038995 0.81 ALDH1A1 (0.52) SGMS2NPC1PKMRAB9AALDH1A1
SCHEMBL8039098 0.81 HPGD (0.48) TRPM8NPC1RAB9AALDH1A1MEN1
SCHEMBL8025478 0.81 APP (0.51) TRPM8NPC1RAB9AMEN1KMT2A
SCHEMBL8041684 0.80 SMPD1 (0.44) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL8025483 0.79 MEN1 (0.46) SGMS2NPC1PKMRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed