SCHEMBL8035618

SCHEMBL8035618

COc1cc(C(F)(F)F)c(C(=O)NC(=O)N(C)C2CC2)cc1OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
PKM P14618 1/20 0.43
SMPD1 P17405 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CTSV O60911 2/20 0.40
CTSL P07711 2/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
SMO Q99835 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SRD5A1 P18405 1/20 0.39
SRD5A2 P31213 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025472 0.95 SGMS2 (0.42) APPNPC1RAB9APKMSMPD1
SCHEMBL8025476 0.89 SMPD1 (0.47) APPNPC1RAB9ASMPD1HDAC1
SCHEMBL8041224 0.87 SMPD1 (0.44) APPNPC1RAB9APKMSMPD1
SCHEMBL8041684 0.87 SMPD1 (0.44) APPNPC1RAB9ASMPD1HDAC1
SCHEMBL8025478 0.85 APP (0.51) APPNPC1RAB9ASMPD1HDAC1
SCHEMBL8035586 0.85 SMPD1 (0.45) APPNPC1RAB9ASMPD1HDAC1
SCHEMBL8035110 0.84 TRPM8 (0.45) APPNPC1RAB9APKMSMPD1
SCHEMBL8025483 0.84 MEN1 (0.46) APPNPC1RAB9APKMSMPD1
SCHEMBL8038995 0.82 ALDH1A1 (0.52) NPC1RAB9APKMSMPD1HDAC1
SCHEMBL8037062 0.82 SMPD1 (0.51) NPC1RAB9ASMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed