SCHEMBL8041228

SCHEMBL8041228

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NC2CCCCC2)cc1OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 1/20 0.53
ALDH1A1 P00352 3/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
CNR2 P34972 2/20 0.45
CNR1 P21554 1/20 0.45
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SMPD1 P17405 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
EPHX1 P07099 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
PPIA P62937 1/20 0.43
APP P05067 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8038995 0.99 ALDH1A1 (0.52) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8025483 0.95 MEN1 (0.46) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8039003 0.92 CNR1 (0.47) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8035606 0.87 SGMS2 (0.56) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8037216 0.86 SGMS2 (0.58) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8035583 0.86 SGMS2 (0.58) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8025472 0.85 SGMS2 (0.42) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8039098 0.84 HPGD (0.48) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL8035613 0.83 S1PR1 (0.54) SGMS2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8025544 0.83 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed