SCHEMBL8037259

SCHEMBL8037259

CC(C)(C)OC(=O)N1CCCC(c2cnc[nH]2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.49
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
ALDH1A1 P00352 2/20 0.46
GLA P06280 1/20 0.46
RECQL P46063 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MAPT P10636 2/20 0.44
THRB P10828 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
USP30 Q70CQ3 1/20 0.43
CYP2C9 P11712 1/20 0.42
CCNK O75909 1/20 0.42
CDK12 Q9NYV4 1/20 0.42
GPR119 Q8TDV5 2/20 0.41
TRPV3 Q8NET8 1/20 0.41
FPR2 P25090 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9986456 0.78 HPGDS (0.49) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL9986181 0.77 HPGDS (0.50) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL9293554 0.77 HPGDS (0.50) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL26667052 0.76 PDE4B (0.52) HPGDSJAK2JAK1HPGDALDH1A1
SCHEMBL25343613 0.76 PDE4B (0.52) HPGDSJAK2JAK1HPGDALDH1A1
SCHEMBL9986338 0.76 JAK2 (0.55) JAK2JAK1MEN1KMT2AUSP30
SCHEMBL20284612 0.76 CYP2C9 (0.63) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL20284463 0.76 CYP2C9 (0.54) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL23124118 0.76 HPGDS (0.49) HPGDSJAK2JAK1KDM4EHPGD
SCHEMBL15551483 0.76 HPGDS (0.54) HPGDSJAK2JAK1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000076514-A1 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-12-21 WO disclosed